Arimidex (anastrozole) – tablets products “antiaromatase” which is used by many bodybuilders to prevent gynecomastia and edema – side effects associated with testosterone esters.
Anastrozole – the most popular are guaranteed a quick way to get rid of aroma and its effects early on. Is more effective than other drugs known antiaromataznyh such as tamoxifen or Nolvadex.
Aromatase – a key enzyme in the biosynthesis of estrogen.
Anastrozole reduce aromatase activity by approximately 95% from baseline.
Anastrozole has a specific activity of aromatase inhibition, in contrast with megestrol acetate or aminoglutethimide.
Anastrozole has no effect on adrenal steroidogenesis.
Anastrozole can effectively suppress high aromatization. The drug is rapidly and completely absorbed from the gastrointestinal tract, maximum concentration of drug in the blood is reached after 2 hours of fasting, is metabolized slowly and therefore has a relatively long half-life (40-50 hours) from the mainly in urine and to a lesser extent – quantities bile.
One should use the drug once a day for 1 mg (1 tablet). The effect is completely reached after 10-14 days of starting treatment.
Do not take more than 1 Anastrozole tablets per day, and a long time.