Type: Anastrazolum Tablets/1 mg
Arimidex (Anastrozole) – tableted product “antiaromatase” which is used by many bodybuilders to prevent gynecomastia and edema – side effects associated with the use of testosterone esters. Anastrozole – the most popular are guaranteed a quick way to get rid of flavor and its effects early on. Is much more effective than other known antiaromataznyh drugs such as Tamoxifen or Nolvadex. Aromatase – a key enzyme of estrogen biosynthesis.Anastrozole reduces aromatase activity by approximately 95% from baseline.Anastrozole has a specific inhibitory activity of aromatase, in contrast to megestrol acetate or aminoglutethimide.Anastrozole has no effect on adrenal steroidogenesis.Anastrozole can effectively suppress the high aromatization. The drug is rapidly and completely absorbed from the gastrointestinal tract, the maximum concentration of drug in the blood is reached after 2 h after fasting, is metabolized slowly and therefore has a relatively long half-life (40-50 hours), derived mainly from the urine and to a lesser quantities – the bile. One should use the drug once a day for 1 mg (1 tablet). The effect is completely achieved after 10-14 days after the start of treatment. Do not take more than 1 Anastrozole tablets a day, as well as a long time.